Providing a handy reference to synthetic methods and practical techniques, Heterocyclic Chemistry in Drug Discovery fuses heterocyclic chemistry and drug discovery, two areas that have gone hand-in-hand in the practice of medicinal chemistry, but have not yet come together for training novice medicinal chemists and students. Rich with numerous case studies to illustrate the real-world drug discovery applications, this book brings together the collective 100-plus years of drug discovery experience from academic and industry contributors to provide valuable insight into the role and application of heterocyclic chemistry for pharmaceuticals.